SCHEMBL7805535

SCHEMBL7805535

COc1ccc(COC(=O)N2C[C@@H](S)C[C@H]2CNS(=O)(=O)NCCO)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.40
HTT P42858 2/20 0.38
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MMP1 P03956 3/20 0.37
MMP3 P08254 3/20 0.37
MMP7 P09237 3/20 0.37
MMP9 P14780 3/20 0.37
MMP13 P45452 2/20 0.37
ALDH1A1 P00352 2/20 0.36
NPSR1 Q6W5P4 1/20 0.35
TP53 P04637 1/20 0.35
P2RX4 Q99571 1/20 0.35
ECE1 P42892 1/20 0.35
MMP2 P08253 1/20 0.35
MMP8 P22894 1/20 0.35
ITGB3 P05106 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGAV P06756 1/20 0.34
ITGA2B P08514 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7800322 0.88 CA1 (0.43) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7811557 0.88 CA1 (0.43) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7805565 0.87 CA12 (0.41) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7806813 0.83 CHRM1 (0.37) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7807913 0.83 CHRM1 (0.37) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7800300 0.79 P2RX4 (0.42) GRIN2BHTTPKMSMN1; SMN2ALDH1A1
SCHEMBL7805534 0.78 MMP1 (0.37) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7805575 0.77 PKM (0.38) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7800321 0.77 PKM (0.38) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7806890 0.76 CA12 (0.42) GRIN2BHTTPKMSMN1; SMN2MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed