SCHEMBL7805565

SCHEMBL7805565

COc1ccc(COC(=O)N2C[C@@H](S)C[C@H]2CNS(N)(=O)=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA5A P35218 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
GRIN2B Q13224 1/20 0.40
HTT P42858 2/20 0.40
PKM P14618 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MMP1 P03956 2/20 0.39
MMP3 P08254 2/20 0.39
MMP7 P09237 2/20 0.39
MMP9 P14780 2/20 0.39
MMP13 P45452 1/20 0.39
ALDH1A1 P00352 4/20 0.38
NPSR1 Q6W5P4 1/20 0.38
P2RX4 Q99571 1/20 0.38
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7806890 0.89 CA12 (0.42) CA12CA1CA2CA5ACA9
SCHEMBL7811557 0.87 CA1 (0.43) CA1CA2GRIN2BHTTPKM
SCHEMBL7800322 0.87 CA1 (0.43) CA1CA2GRIN2BHTTPKM
SCHEMBL7805535 0.87 GRIN2B (0.40) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7806813 0.86 CHRM1 (0.37) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7807913 0.86 CHRM1 (0.37) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7809178 0.85 CA12 (0.39) CA12CA1CA2CA5ACA9
SCHEMBL195204 0.85 CA12 (0.40) CA12CA1CA2CA9ALDH1A1
SCHEMBL195205 0.85 CA12 (0.40) CA12CA1CA2CA9ALDH1A1
SCHEMBL7809302 0.85 CA12 (0.38) CA12CA1CA2CA5ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed