SCHEMBL7806465

SCHEMBL7806465

Nc1nc(SC(c2ccccc2)c2ccccc2)c2[nH]cnc2n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.60
POLB P06746 1/20 0.60
CYP1A2 P05177 6/20 0.59
CYP3A4 P08684 5/20 0.59
CYP2C19 P33261 5/20 0.59
CYP2D6 P10635 4/20 0.59
CYP2C9 P11712 3/20 0.59
NUDT1 P36639 2/20 0.59
ALDH1A1 P00352 1/20 0.59
TOP2A P11388 1/20 0.59
HPGD P15428 1/20 0.59
HIF1A Q16665 1/20 0.59
HSD17B10 Q99714 1/20 0.59
MAP3K5 Q99683 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.55
ENPP1 P22413 1/20 0.51
CDK1 P06493 5/20 0.48
CDK2 P24941 5/20 0.48
CCNB1 P14635 4/20 0.48
CCNA2 P20248 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7806463 0.78 PIN1 (0.39) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL2115657 0.75 PIN1 (1.00) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL24846512 0.74 CYP1A2 (1.00) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL7674651 0.74 CYP1A2 (0.77) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL9346526 0.74 MAP3K5 (0.72) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL94363 0.72 MAP3K5 (1.00) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL24846509 0.71 CYP1A2 (0.88) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL24846960 0.71 CYP1A2 (1.00) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL6318896 0.70 MAP3K5 (0.61) PIN1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL24846433 0.70 CYP1A2 (0.79) PIN1POLBCYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0352953-B1 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 2001-01-03 EP disclosed
US-5017701-A Process for the preparation of purine derivatives BEECHAM GROUP, P.L.C. (GB) 1991-05-21 US disclosed
EP-0352953-A2 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 1990-01-31 EP disclosed