SCHEMBL7806477

SCHEMBL7806477

CS(=O)(=O)Nc1cc(N)ccc1Br

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.42
SLC22A12 Q96S37 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
KEAP1 Q14145 3/20 0.38
NFE2L2 Q16236 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PIK3CD O00329 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
HTR6 P50406 1/20 0.36
PTGS1 P23219 3/20 0.36
PTGS2 P35354 3/20 0.36
ADRB3 P13945 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244812 0.82 L3MBTL1 (0.42) L3MBTL1CA12CA1CA2CA9
SCHEMBL1290875 0.79 KEAP1 (0.43) BACE1SLC22A12CA1CA2CA9
SCHEMBL2336547 0.79 CCNT1 (0.49) BACE1L3MBTL1KEAP1NFE2L2ALDH1A1
SCHEMBL30764888 0.79 KEAP1 (0.43) BACE1SLC22A12CA1CA2CA9
SCHEMBL23226730 0.78 ADRB3 (0.56) ADRB3
SCHEMBL18332101 0.78 KDM1A (0.51) L3MBTL1KEAP1NFE2L2PIK3CDPIK3CA
SCHEMBL5202983 0.78 PIK3CD (0.47) BACE1L3MBTL1ALDH1A1PIK3CDPIK3CA
SCHEMBL19099945 0.77 GAA (0.41) L3MBTL1KEAP1NFE2L2ALDH1A1PIK3CD
Ammonia Solution, Strong SCHEMBL2211253 0.76 KDM1A (0.50) L3MBTL1KEAP1NFE2L2PIK3CDPIK3CA
SCHEMBL2310180 0.76 PTGS1 (0.42) L3MBTL1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010143664-A1 TETRACYCLIC COMPOUND 中外製薬株式会社 (JP) 2010-12-16 WO disclosed