SCHEMBL1290875

SCHEMBL1290875

Cc1ccc(Br)c(NS(C)(=O)=O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
BACE1 P56817 1/20 0.43
PARP14 Q460N5 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
NR3C1 P04150 1/20 0.41
PTGS1 P23219 3/20 0.41
PTGS2 P35354 2/20 0.41
SLC22A12 Q96S37 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30764888 1.00 KEAP1 (0.43) KEAP1NFE2L2BACE1PARP14SMN1; SMN2
SCHEMBL1290883 0.85 KMT2A (0.49) KEAP1NFE2L2SMN1; SMN2NPC1LMNA
SCHEMBL13303941 0.82 PTGS1 (0.47) KEAP1NFE2L2PARP14NPC1LMNA
SCHEMBL13842603 0.80 KMT2A (0.51) KEAP1NFE2L2PARP14NPC1POLB
SCHEMBL7806477 0.79 BACE1 (0.42) KEAP1NFE2L2BACE1PTGS1PTGS2
SCHEMBL12900927 0.77 MEN1 (0.49) KEAP1NFE2L2BACE1PARP14NPC1
SCHEMBL19420697 0.77 TP53 (0.45) KEAP1NFE2L2PARP14SMN1; SMN2NPC1
SCHEMBL14014069 0.77 KDM1A (0.49) KEAP1NFE2L2PARP14NPC1LMNA
SCHEMBL13393229 0.77 ADRA2A (0.57) PARP14SMN1; SMN2CA1CA2CA9
SCHEMBL4792308 0.77 MAPK1 (0.49) SMN1; SMN2LMNANR3C1PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111836801-B Compounds for inhibiting TNIK and medical use thereof 韩国化学硏究院 2024-02-02 CN disclosed
CN-111836801-A Compound for inhibiting TNIK and medical application thereof 韩国化学硏究院 2020-10-27 CN disclosed
WO-2012045194-A1 BENZODIAZEPINONES AS FAK INHIBITORS FOR TREATMENT OF CANCER ABBOTT LABORATORIES (US) 2012-04-12 WO disclosed