SCHEMBL7806909

SCHEMBL7806909

CCCCOC(=O)N=C(N)c1ccc(NCC#Cc2cc(C)c(C(=O)N3CCCC3)cc2C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
HPGD P15428 6/20 0.38
SMN1; SMN2 Q16637 5/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
NR1I2 O75469 1/20 0.35
F2 P00734 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
SLC6A2 P23975 1/20 0.35
AGTR1 P30556 1/20 0.35
SLC6A3 Q01959 1/20 0.35
SCN5A Q14524 1/20 0.35
RAB9A P51151 6/20 0.34
NPC1 O15118 5/20 0.34
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7806927 0.91 HPGD (0.41) ALDH1A1HPGDSMN1; SMN2KMT2AMEN1
SCHEMBL7806863 0.88 HRH3 (0.35) ALDH1A1HPGDKMT2AMEN1NR1I2
SCHEMBL7799453 0.84 HPGD (0.39) ALDH1A1HPGDSMN1; SMN2KMT2AMEN1
SCHEMBL7804882 0.83 HPGD (0.38) ALDH1A1HPGDSMN1; SMN2KMT2AMEN1
SCHEMBL7806159 0.83 ALDH1A1 (0.36) ALDH1A1HPGDSMN1; SMN2KMT2AMEN1
SCHEMBL7809959 0.82 SMN1; SMN2 (0.39) ALDH1A1SMN1; SMN2KMT2ANR1I2F2
SCHEMBL7806169 0.80 NR1I2 (0.34) ALDH1A1KMT2AMEN1NR1I2F2
SCHEMBL6563662 0.80 F10 (0.41) HPGDKMT2AMEN1F2
SCHEMBL7809950 0.79 PIK3CA (0.40) ALDH1A1SMN1; SMN2NR1I2F2ADORA3
SCHEMBL7806152 0.78 HRH3 (0.37) ALDH1A1NR1I2F2ADORA3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM KG (DE) 2001-10-10 EP disclosed
WO-2000035859-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-06-22 WO disclosed