SCHEMBL7807876

SCHEMBL7807876

CCC(=C(c1ccc(O)cc1)c1ccc(OCCN2CCCC2)cc1)c1ccccc1

nearest known ligand 0.91

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.91
PSMB1 P20618 6/20 0.91
PSMB5 P28074 5/20 0.91
PSMB2 P49721 2/20 0.91
ESR2 Q92731 2/20 0.81
PDE1A P54750 2/20 0.81
PDE1B Q01064 2/20 0.81
PDE1C Q14123 2/20 0.81
ESRRG P62508 4/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17151967 1.00 ESR1 (0.91) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL24505428 1.00 ESR1 (0.91) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL29822053 0.95 PSMB1 (1.00) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL15648408 0.95 PSMB1 (1.00) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL23266922 0.95 ESR1 (0.81) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL7650153 0.95 PSMB1 (1.00) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL30902018 0.95 PSMB1 (1.00) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL7650156 0.95 PSMB1 (1.00) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL23266947 0.90 ESR1 (0.90) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL24354598 0.90 ESR1 (0.82) ESR1PSMB1PSMB5PSMB2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1127045-A2 USE OF TRIPHENYLBUTENE DERIVATIVES FOR THE TREATMENT OF NEUROLOGICAL DISORDERS AstraZeneca AB (SE) 2001-08-29 EP claimed
WO-2000025767-A2 USE OF TRIPHENYLBUTENE DERIVATIVES FOR THE TREATMENT OF NEUROLOGICAL DISORDERS ASTRAZENECA AB (SE) 2000-05-11 WO claimed