SCHEMBL7808570

SCHEMBL7808570

Clc1ccc(-c2nc(I)c[nH]2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.45
CXCR2 P25025 1/20 0.44
TYMP P19971 1/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HRH1 P35367 1/20 0.41
KMO O15229 4/20 0.40
NOTUM Q6P988 2/20 0.40
CYP1B1 Q16678 1/20 0.39
IDO1 P14902 1/20 0.39
MAPK13 O15264 1/20 0.38
RAF1 P04049 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
NPY5R Q15761 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4658269 0.81 KMO (0.40) AHRCXCR2TYMPNPC1RAB9A
SCHEMBL4658006 0.80 AHR (0.37) AHRCXCR2TYMPNPC1RAB9A
SCHEMBL4657944 0.78 KDM4E (0.40) TYMPNPC1RAB9ANOTUM
SCHEMBL3130583 0.75 CXCR2 (0.48) AHRCXCR2NPC1RAB9AKMO
SCHEMBL2552851 0.75 TYMP (0.41) AHRCXCR2TYMPNPC1RAB9A
SCHEMBL11014522 0.73 TYMP (0.40) AHRCXCR2TYMPNPC1RAB9A
SCHEMBL31305411 0.72 MAPK13 (0.49) AHRCXCR2NPC1RAB9AKMO
SCHEMBL2944949 0.72 MAPK13 (0.49) AHRCXCR2NPC1RAB9AKMO
SCHEMBL11545138 0.72 CA12 (0.44) AHRCXCR2TYMPNPC1RAB9A
SCHEMBL1719052 0.71 AHR (0.45) AHRCXCR2TYMPNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed