SCHEMBL7809186

SCHEMBL7809186

COc1ccc(COC(=O)N2C[C@@H](SC(C)=O)C[C@H]2CN2C(=O)c3ccccc3C2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 2/20 0.39
P2RX4 Q99571 1/20 0.39
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 2/20 0.38
POLB P06746 1/20 0.38
APEX1 P27695 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
RPS6KA2 Q15349 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
GRIN2B Q13224 1/20 0.37
APAF1 O14727 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
MMP2 P08253 1/20 0.37
MMP9 P14780 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811581 0.87 ATM (0.41) ALDH1A1HSD17B10TDP1
SCHEMBL7806847 0.86 POLB (0.38) CASP3NPC1GAAP2RX4ALDH1A1
SCHEMBL7805553 0.86 CASP3 (0.43) CASP3NPC1GAAP2RX4ALDH1A1
SCHEMBL7811563 0.81 NPSR1 (0.46) CASP3ALDH1A1POLB
SCHEMBL7805526 0.81 CASP3 (0.41) CASP3NPC1GAAP2RX4ALDH1A1
SCHEMBL7800302 0.81 ECE1 (0.37) NPC1ALDH1A1MEN1KMT2A
SCHEMBL7809302 0.77 CA12 (0.38) P2RX4ALDH1A1GRIN2BMMP2MMP9
SCHEMBL8572110 0.75 POLB (0.49) NPC1POLB
SCHEMBL10391482 0.75 GAA (0.49) GAAALDH1A1
SCHEMBL9202926 0.74 POLB (0.46) NPC1ALDH1A1POLBTDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed