SCHEMBL7806847

SCHEMBL7806847

COc1ccc(COC(=O)N2C[C@@H](SC(c3ccccc3)(c3ccccc3)c3ccccc3)C[C@H]2CN2C(=O)c3ccccc3C2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
APEX1 P27695 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CASP3 P42574 1/20 0.37
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37
ALDH1A1 P00352 3/20 0.37
MMP2 P08253 1/20 0.37
MMP9 P14780 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
P2RX4 Q99571 1/20 0.37
TP53 P04637 1/20 0.37
RPS6KA2 Q15349 1/20 0.36
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7809185 0.87 TDP1 (0.41) TDP1ALDH1A1
SCHEMBL7805486 0.87 P2RX4 (0.41) ALDH1A1MMP9NPSR1P2RX4TP53
SCHEMBL7809186 0.86 CASP3 (0.40) POLBAPEX1HSD17B10TDP1CASP3
SCHEMBL7805571 0.86 KIF11 (0.40) NPC1ALDH1A1MMP9NPSR1P2RX4
Acetic Acid SCHEMBL7809331 0.84 ALDH1A1 (0.39) ALDH1A1MMP9NPSR1P2RX4TP53
SCHEMBL7805553 0.83 CASP3 (0.43) POLBAPEX1HSD17B10TDP1CASP3
SCHEMBL7809176 0.83 HCRTR2 (0.41) ALDH1A1MMP2MMP9NPSR1P2RX4
SCHEMBL7811618 0.81 ALDH1A1 (0.42) POLBALDH1A1MMP2MMP9NPSR1
SCHEMBL7805536 0.79 CA1 (0.43) ALDH1A1MMP2MMP9NPSR1TP53
SCHEMBL7800320 0.79 MMP1 (0.38) POLBALDH1A1MMP2MMP9NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed