SCHEMBL7811563

SCHEMBL7811563

C=CCOC(=O)N1C[C@@H](SC(C)=O)C[C@H]1CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.46
ALDH1A1 P00352 4/20 0.35
ECE1 P42892 1/20 0.35
CYP19A1 P11511 1/20 0.35
POLB P06746 1/20 0.34
FAAH O00519 3/20 0.34
MGLL Q99685 1/20 0.34
ELANE P08246 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
RHOA P61586 1/20 0.32
PLIN1 O60240 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
PLIN5 Q00G26 1/20 0.32
ABHD5 Q8WTS1 1/20 0.32
CASP3 P42574 1/20 0.32
F2 P00734 1/20 0.32
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9132827 0.89 NPSR1 (0.43) NPSR1ALDH1A1CYP19A1POLBFAAH
SCHEMBL7800302 0.84 ECE1 (0.37) ALDH1A1ECE1PLIN1MAPTHPGD
SCHEMBL7809186 0.81 CASP3 (0.40) ALDH1A1POLBCASP3
SCHEMBL7811591 0.80 NPSR1 (0.45) NPSR1ALDH1A1CYP19A1POLBFAAH
SCHEMBL7811581 0.79 ATM (0.41) ALDH1A1MAPTHPGD
SCHEMBL7805577 0.79 ECE1 (0.33) ECE1CYP19A1SIGMAR1
SCHEMBL9215991 0.78 ECE1 (0.34) ALDH1A1ECE1CYP19A1POLBFAAH
SCHEMBL8833259 0.78 ECE1 (0.34) ALDH1A1ECE1CYP19A1POLBFAAH
SCHEMBL7852448 0.77 ECE1 (0.37) ALDH1A1ECE1CYP19A1ELANESIGMAR1
SCHEMBL9461797 0.77 ECE1 (0.34) ECE1CYP19A1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed