SCHEMBL7809666

SCHEMBL7809666

OCc1nc2cc(Sc3ccnc4cc(C(F)(F)F)ccc34)ccc2[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.36
NCF1 P14598 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SLC22A12 Q96S37 1/20 0.35
KIF11 P52732 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
PARP1 P09874 1/20 0.34
KDR P35968 4/20 0.34
PRKD3 O94806 2/20 0.34
MAP4K4 O95819 2/20 0.34
GSK3A P49840 2/20 0.34
GSK3B P49841 2/20 0.34
AURKB Q96GD4 2/20 0.34
PRKD2 Q9BZL6 2/20 0.34
CLK4 Q9HAZ1 2/20 0.34
PDE10A Q9Y233 1/20 0.34
MARK3 P27448 1/20 0.34
MAPKAPK2 P49137 1/20 0.34
PRKCZ Q05513 1/20 0.34
PRKAA1 Q13131 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7809674 0.92 TDP1 (0.40) ADRB2NCF1ALDH1A1SLC22A12KDR
SCHEMBL4556153 0.80 TDP1 (0.47) KIF11PDE10AKDM4ETDP1
SCHEMBL8565612 0.73 MEN1 (0.48) ADRB2NCF1ALDH1A1SLC22A12KIF11
SCHEMBL2015868 0.71 TDP1 (0.44) ALDH1A1KDM4EFGFR1TDP1
SCHEMBL8565482 0.70 ADRB2 (0.42) ADRB2NCF1ALDH1A1SLC22A12PARP1
SCHEMBL7808588 0.70 TDP1 (0.43) ALDH1A1PRKD3AURKBCLK4TAOK1
SCHEMBL9597974 0.70 PDE10A (0.47) PDE10AKDM4E
Hydrochloric Acid SCHEMBL8480475 0.69 TDP1 (0.42) ALDH1A1PRKD3AURKBCLK4TAOK1
SCHEMBL7808616 0.69 NPC1 (0.50) ALDH1A1L3MBTL1TDP1
SCHEMBL7808661 0.69 TDP1 (0.43) ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820990-B1 Benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR (FR) 2001-01-17 EP disclosed
US-5972968-A INTERLEUKIN INHIBITOR ADIR ET COMPAGNIE (FR) 1999-10-26 US disclosed
EP-0820990-A2 Novel benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR ET COMPAGNIE (FR) 1998-01-28 EP disclosed