SCHEMBL7811858

SCHEMBL7811858

Cc1ccccc1-c1nc2c(o1)C(=O)c1ccccc1C2=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP1 O94782 4/20 0.67
USP19 O94966 2/20 0.67
WDR48 Q8TAF3 1/20 0.67
UCHL3 P15374 1/20 0.60
USP2 O75604 2/20 0.57
USP8 P40818 2/20 0.57
OTUB1 Q96FW1 2/20 0.57
USP36 Q9P275 1/20 0.57
RAB9A P51151 6/20 0.49
NPC1 O15118 6/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
CASP3 P42574 2/20 0.49
SENP8 Q96LD8 2/20 0.49
SENP7 Q9BQF6 2/20 0.49
SENP6 Q9GZR1 2/20 0.49
NOTUM Q6P988 1/20 0.47
ELANE P08246 1/20 0.46
IKBKB O14920 1/20 0.46
F7 P08709 1/20 0.45
F3 P13726 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21498209 0.86 USP1 (0.64) USP1USP19WDR48UCHL3USP2
SCHEMBL7968066 0.81 USP1 (0.77) USP1USP19WDR48UCHL3USP2
SCHEMBL7808221 0.81 USP1 (0.67) USP1USP19WDR48UCHL3USP2
SCHEMBL7808123 0.81 USP1 (0.68) USP1USP19WDR48UCHL3USP2
SCHEMBL29629184 0.80 USP1 (1.00) USP1USP19WDR48UCHL3USP2
SCHEMBL7808226 0.80 USP1 (1.00) USP1USP19WDR48UCHL3USP2
SCHEMBL29629183 0.80 USP1 (1.00) USP1USP19WDR48UCHL3USP2
SCHEMBL7818903 0.80 USP1 (0.60) USP1USP19WDR48UCHL3USP2
SCHEMBL7812967 0.78 USP1 (0.71) USP1USP19WDR48UCHL3USP2
SCHEMBL19220486 0.77 USP1 (0.82) USP1USP19WDR48UCHL3USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0876356-B1 USE OF TRICYCLIC 1,4-DIHYDRO-1,4-DIOXO-1H-NAPHTHALENE DERIVATIVES, RESULTING NOVEL COMPOUNDS AND THERAPEUTICAL USE THEREOF INNOTHERA SA LAB (FR) 2001-10-31 EP claimed
US-10450281-B1 Compounds and methods for treating cancer DANA-FARBER CANCER INSTITUTE, INC. (US) 2019-10-22 US disclosed
US-6262095-B1 TREATMENT OF ILLNESS ASSOCIATED WITH AN ALTERATION IN VENOUS FUNCTION AND/OR INFLAMMATORY EDEMA LABORATOIRE INNOTHERA (FR) 2001-07-17 US disclosed
EP-0876356-A1 USE OF TRICYCLIC 1,4-DIHYDRO-1,4-DIOXO-1H-NAPHTHALENE DERIVATIVES, RESULTING NOVEL COMPOUNDS AND THERAPEUTICAL USE THEREOF LABORATOIRE INNOTHERA Société Anonyme (FR) 1998-11-11 EP disclosed
WO-1997021684-A1 USE OF TRICYCLIC 1,4-DIHYDRO-1,4-DIOXO-1H-NAPHTHALENE DERIVATIVES, RESULTING NOVEL COMPOUNDS AND THERAPEUTICAL USE THEREOF LABORATOIRE INNOTHERA, SOCIETE ANONYME (FR) 1997-06-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10450281-B1 Compounds and methods for treating cancer USP8, USP2, NEDD8 USP1 7/4885USP19 22/4885WDR48 306/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.