SCHEMBL7812401

SCHEMBL7812401

COC(=O)c1[nH]c(C(C)(C)C)cc1CN

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.48
RAF1 P04049 2/20 0.47
LOXL2 Q9Y4K0 2/20 0.37
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
USP2 O75604 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
KIF11 P52732 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3220088 0.79 MAPK14 (0.55) MAPK14RAF1KDM4EALDH1A1GAA
SCHEMBL13487957 0.73 MAPK14 (0.52) MAPK14RAF1KDM4EALDH1A1GAA
SCHEMBL10308264 0.73 MAPK14 (0.49) MAPK14RAF1KDM4EALDH1A1GAA
SCHEMBL3220272 0.71 MAPK14 (0.47) MAPK14RAF1ALDH1A1NPSR1MAPT
SCHEMBL16240346 0.68 LMNA (0.42) MAPK14RAF1KDM4EALDH1A1GAA
SCHEMBL3539674 0.67 MAPK14 (0.52) MAPK14RAF1ALDH1A1NPSR1USP2
SCHEMBL10717450 0.67 MAPT (0.49) MAPK14RAF1KDM4EALDH1A1GAA
SCHEMBL4423633 0.66 MAPK14 (0.51) MAPK14RAF1KDM4EALDH1A1GAA
SCHEMBL13315128 0.66 MAPK14 (0.49) MAPK14RAF1KDM4EALDH1A1GAA
SCHEMBL5775175 0.66 ALDH1A1 (0.46) MAPK14RAF1KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986382-A4 RAF KINASE INHIBITORS BAYER AG (US) 2001-04-11 EP disclosed
EP-0986382-A1 RAF KINASE INHIBITORS Bayer Corporation (US) 2000-03-22 EP disclosed
WO-1998052559-A1 RAF KINASE INHIBITORS BAYER CORPORATION (US) 1998-11-26 WO disclosed