SCHEMBL7812427

SCHEMBL7812427

CN1CCCN(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHKA P35790 8/20 0.68
KDM4E B2RXH2 5/20 0.54
ALDH1A1 P00352 4/20 0.54
POLB P06746 1/20 0.54
CA2 P00918 1/20 0.53
NCF1 P14598 1/20 0.53
PRMT6 Q96LA8 1/20 0.53
CASP1 P29466 1/20 0.52
CASP5 P51878 1/20 0.52
GAA P10253 1/20 0.51
CYP3A4 P08684 3/20 0.50
CYP2D6 P10635 3/20 0.50
HTR7 P34969 1/20 0.49
USP2 O75604 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C19 P33261 1/20 0.49
MEN1 O00255 1/20 0.49
TP53 P04637 1/20 0.49
KMT2A Q03164 1/20 0.49
MAPT P10636 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10819405 0.94 CHKA (0.57) CHKAKDM4EALDH1A1CASP1CASP5
SCHEMBL8974017 0.90 ALDH1A1 (0.60) CHKAKDM4EALDH1A1CASP1CASP5
SCHEMBL18783072 0.88 ALDH1A1 (0.56) CHKAKDM4EALDH1A1POLBCASP1
SCHEMBL6028265 0.85 ALDH1A1 (0.67) KDM4EALDH1A1CASP1CASP5GAA
SCHEMBL2056180 0.84 CHKA (0.91) CHKAKDM4EALDH1A1POLBCA2
SCHEMBL428016 0.84 CHKA (0.52) CHKAKDM4EALDH1A1CASP1CASP5
SCHEMBL6925369 0.84 CHKA (0.52) CHKAKDM4EALDH1A1CASP1CASP5
SCHEMBL31010361 0.83 ALDH1A1 (0.70) KDM4EALDH1A1CASP1CASP5GAA
SCHEMBL29777509 0.83 LMNA (0.53) CHKAKDM4EALDH1A1CA2NCF1
SCHEMBL545449 0.83 LMNA (0.53) CHKAKDM4EALDH1A1CA2NCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140880-A1 HOMOPIPERAZINE DERIVATIVES AS SELECTIVE EMOPAMIL INHIBITORS AstraZeneca AB (SE) 2001-10-10 EP claimed
WO-2000039110-A1 HOMOPIPERAZINE DERIVATIVES AS SELECTIVE EMOPAMIL INHIBITORS ASTRAZENECA AB (SE) 2000-07-06 WO claimed
EP-1140880-A1 HOMOPIPERAZINE DERIVATIVES AS SELECTIVE EMOPAMIL INHIBITORS AstraZeneca AB (SE) 2001-10-10 EP disclosed
WO-2000039110-A1 HOMOPIPERAZINE DERIVATIVES AS SELECTIVE EMOPAMIL INHIBITORS ASTRAZENECA AB (SE) 2000-07-06 WO disclosed