SCHEMBL8974017

SCHEMBL8974017

FC(F)(F)c1cc(CN2CCCN(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)CCN(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)CCCN(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)CC2)cc(C(F)(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.60
KDM4E B2RXH2 2/20 0.60
CASP1 P29466 1/20 0.60
CASP5 P51878 1/20 0.60
GAA P10253 1/20 0.60
CYP2D6 P10635 7/20 0.58
CYP3A4 P08684 7/20 0.58
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
TP53 P04637 1/20 0.56
CHKA P35790 1/20 0.53
USP2 O75604 4/20 0.52
CYP2C19 P33261 3/20 0.52
CYP1A2 P05177 2/20 0.52
TSHR P16473 6/20 0.51
CYP2C9 P11712 2/20 0.50
HPGD P15428 1/20 0.48
LMNA P02545 1/20 0.46
HIF1A Q16665 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6028265 0.94 ALDH1A1 (0.67) ALDH1A1KDM4ECASP1CASP5GAA
SCHEMBL31010361 0.92 ALDH1A1 (0.70) ALDH1A1KDM4ECASP1CASP5GAA
SCHEMBL7812427 0.90 CHKA (0.68) ALDH1A1KDM4ECASP1CASP5GAA
SCHEMBL17048623 0.87 ALDH1A1 (0.59) ALDH1A1KDM4ECASP1CASP5GAA
SCHEMBL8974312 0.86 USP2 (0.52) ALDH1A1KDM4ECASP1CASP5GAA
SCHEMBL8973698 0.86 USP2 (0.52) ALDH1A1KDM4ECASP1CASP5GAA
SCHEMBL24565989 0.86 ALDH1A1 (0.54) ALDH1A1KDM4ECASP1CASP5GAA
SCHEMBL4935986 0.86 ALDH1A1 (0.54) ALDH1A1KDM4ECASP1CASP5GAA
SCHEMBL10819405 0.85 CHKA (0.57) ALDH1A1KDM4ECASP1CASP5GAA
SCHEMBL19625264 0.85 CYP2D6 (0.55) ALDH1A1KDM4ECASP1CASP5GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536491-A 19 F poly aza macrocyclic MRI contrast medium TERUMO KABUSHIKI KAISHA (JP) 1996-07-16 US disclosed
EP-0628316-A1 19F-MRI contrast medium, having a macrocyclic complexant moiety TERUMO KABUSHIKI KAISHA (JP) 1994-12-14 EP disclosed