SCHEMBL7814531

SCHEMBL7814531

CCCNC(=O)c1cc(N)c(NC)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
POLB P06746 1/20 0.52
HPGD P15428 1/20 0.52
HTR4 Q13639 4/20 0.50
CYP1A2 P05177 2/20 0.50
ADRA2A P08913 2/20 0.50
CYP2D6 P10635 2/20 0.50
DRD3 P35462 2/20 0.50
DPP4 P27487 2/20 0.50
HTR3E A5X5Y0 2/20 0.50
HTR3B O95264 2/20 0.50
HTR3A P46098 2/20 0.50
HTR3D Q70Z44 2/20 0.50
HTR3C Q8WXA8 2/20 0.50
SLC22A1 O15245 1/20 0.50
LMNA P02545 1/20 0.50
MPO P05164 1/20 0.50
DRD2 P14416 1/20 0.50
ADRA2C P18825 1/20 0.50
DRD4 P21917 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31215241 0.78 GAA (0.59) ALDH1A1POLBHPGDLMNARAB9A
SCHEMBL1725888 0.78 ALDH1A1 (0.51) ALDH1A1HPGDKMT2A
SCHEMBL1966436 0.78 GAA (0.59) ALDH1A1POLBHPGDLMNARAB9A
Dimethylamine SCHEMBL6109558 0.77 ALDH1A1 (0.64) ALDH1A1POLBHPGDHTR4CYP1A2
SCHEMBL27344771 0.76 ALDH1A1 (0.58) ALDH1A1POLBHPGDHTR4CYP1A2
SCHEMBL19445674 0.74 HTR4 (0.51) ALDH1A1POLBHPGDHTR4CYP1A2
SCHEMBL23261794 0.74 ALDH1A1 (0.50) ALDH1A1POLBHPGDHTR4CYP1A2
SCHEMBL2248029 0.73 ALOX15 (0.43) ALDH1A1HPGD
Hydrochloric Acid SCHEMBL9255163 0.73 MAPT (0.40) ALDH1A1HTR4CYP1A2ADRA2ACYP2D6
SCHEMBL1973112 0.73 ALDH1A1 (0.56) ALDH1A1POLBHPGDCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0794184-B1 6-METHOXY-1H-BENZOTRIAZOLE-5-CARBOXAMIDE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND MEDICINAL COMPOSITION CONTAINING THE SAME DAINIPPON PHARMACEUTICAL CO (JP) 2001-05-30 EP disclosed
US-5932568-A GASTROINTESTINAL DISORDERS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1999-08-03 US disclosed
EP-0794184-A1 6-METHOXY-1H-BENZOTRIAZOLE-5-CARBOXAMIDE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND MEDICINAL COMPOSITION CONTAINING THE SAME DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1997-09-10 EP disclosed