SCHEMBL7816583

SCHEMBL7816583

C1=CC2(CNCCN2)Cc2ccccc21

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.33
HTR2B P41595 1/20 0.33
HTR2A P28223 3/20 0.33
DRD2 P14416 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7825051 0.77 LMNA (0.33) HTR2CHTR2BPARP1
SCHEMBL9124282 0.71 MAPT (0.38) PARP1
SCHEMBL7830015 0.69 HTR2C (0.41) HTR2CHTR2BHTR2ADRD2SLC6A2
SCHEMBL2288761 0.67 PARP1 (0.39) HTR2CHTR2BPARP1
SCHEMBL14760157 0.66 HTR2A (0.39) HTR2CHTR2BHTR2ADRD2SLC6A2
SCHEMBL7830334 0.65 HTR2A (0.33) HTR2CHTR2ADRD2SLC6A2SLC6A4
SCHEMBL258234 0.64 PARP1 (0.36) HTR2CHTR2BPARP1
SCHEMBL1697644 0.64 PARP1 (0.36) HTR2APARP1
SCHEMBL7882155 0.64 PARP1 (0.36) HTR2CHTR2BPARP1
SCHEMBL1725344 0.64 PARP1 (0.36) HTR2CHTR2BPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712845-B1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-17 EP disclosed
US-5633248-A GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS, DIARYLALKYLIDENEDIAMINES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-27 US disclosed
EP-0712845-A1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-22 EP disclosed