SCHEMBL78184

SCHEMBL78184

CCOC(=O)C1C(=O)CCN(C(=O)OCc2ccccc2)C1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.39
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
PARP1 P09874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91294 0.85 PARP1 (0.39) ELANEPDK1PDK2PDK3PDK4
SCHEMBL65230 0.84 MAPT (0.33)
SCHEMBL21235743 0.79 ELANE (0.46) ELANEPARP1
SCHEMBL15185033 0.79 NPC1 (0.43) ELANEPDK1PDK2PDK3PDK4
SCHEMBL66855 0.78 ELANE (0.38) ELANE
SCHEMBL13032699 0.78 ELANE (0.48) ELANEPARP1
SCHEMBL29560191 0.77 SMN1; SMN2 (0.45) ELANEPDK1PDK2PDK3PDK4
SCHEMBL34466974 0.77 PREP (0.42) PDK1PDK2PDK3PDK4
SCHEMBL30781571 0.77 PREP (0.42) PDK1PDK2PDK3PDK4
SCHEMBL78361 0.77 PARP1 (0.43) PDK1PDK2PDK3PDK4PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed