SCHEMBL66855

SCHEMBL66855

CCOC(=O)C1C(c2ccc(O)cc2)CCN(C(=O)OCc2ccccc2)C1CO[Si](C)(C)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.38
TMEM97 Q5BJF2 3/20 0.37
SIGMAR1 Q99720 3/20 0.37
KDM1A O60341 1/20 0.37
RCOR1 Q9UKL0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65686 0.81 PDK1 (0.38) KDM1ARCOR1
SCHEMBL15185033 0.79 NPC1 (0.43) ELANE
SCHEMBL78184 0.78 ELANE (0.39) ELANE
SCHEMBL64035 0.78 SLC6A2 (0.37)
SCHEMBL29560191 0.76 SMN1; SMN2 (0.45) ELANE
SCHEMBL65814 0.76 PPARG (0.39)
SCHEMBL65299 0.75 LTA4H (0.35)
SCHEMBL16080271 0.74 ACE2 (0.40)
SCHEMBL65685 0.73 CHRM5 (0.40) ELANE
SCHEMBL29510871 0.73 PDK1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed