SCHEMBL7818917

SCHEMBL7818917

CCc1cc(C(=O)c2ccoc2Cc2ccc(C)c(C)c2)cc(Br)c1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 3/20 0.41
NR1H4 Q96RI1 2/20 0.34
SLC22A12 Q96S37 5/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
TSHR P16473 2/20 0.33
ESR1 P03372 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
APEX1 P27695 1/20 0.33
MAPK1 P28482 1/20 0.33
ESR2 Q92731 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NCOA1 Q15788 1/20 0.32
NCOA3 Q9Y6Q9 1/20 0.32
HPGD P15428 2/20 0.32
ALOX15 P16050 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6731717 0.72 NR3C1 (0.36) CYP2C19LMNAMAPTNPC1RAB9A
SCHEMBL7674920 0.70 CYP2C19 (0.51) CYP2C19NR1H4SLC22A12LMNAMAPT
SCHEMBL7817806 0.69 KMT2A (0.51) CYP2C19LMNAMAPTPOLBNCOA1
SCHEMBL7670073 0.66 TPMT (0.65) CYP2C19LMNATSHRNCOA1NCOA3
SCHEMBL6740976 0.65 NUDT1 (0.38) ESR1TP53POLBESR2SMN1; SMN2
SCHEMBL24199843 0.62 MAPT (0.51) CYP2C19MAPTL3MBTL1TP53POLB
SCHEMBL21362509 0.61 MAPT (0.45) CYP2C19SLC22A12MAPTTP53HPGD
SCHEMBL24199867 0.61 HTT (0.45) CYP2C19SLC22A12LMNAMAPTTP53
SCHEMBL6736525 0.61 CYP2C19 (0.46) CYP2C19NR1H4LMNAMAPTPOLB
SCHEMBL7670596 0.61 CYP2C19 (0.53) CYP2C19NR1H4SLC22A12LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077968-A1 NAPHTHO[2,3-B]HETEROAR-4-YL DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2001-02-28 EP disclosed
WO-1999058522-A1 NAPHTHO[2,3-B]HETEROAR-4-YL DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1999-11-18 WO disclosed