SCHEMBL7819175

SCHEMBL7819175

COc1ccc(COc2cncc3c2-c2nn(C)c4ccc(NCCN(C)C)c(c24)C3=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 5/20 0.39
NQO1 P15559 2/20 0.37
KAT2B Q92831 2/20 0.37
CYP19A1 P11511 1/20 0.33
CNR2 P34972 2/20 0.32
BCHE P06276 1/20 0.32
RAD52 P43351 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ATM Q13315 1/20 0.32
ACHE P22303 1/20 0.32
SMARCA2 P51531 1/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
CSF1R P07333 1/20 0.31
EHMT2 Q96KQ7 2/20 0.31
MAPT P10636 1/20 0.31
AKT1 P31749 1/20 0.31
RPS6KA1 Q15418 1/20 0.31
PIM1 P11309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7818284 0.93 NQO2 (0.38) NQO2NQO1KAT2BCYP19A1CNR2
SCHEMBL7821158 0.88 TOP2A (0.35) NQO2NQO1CYP19A1CNR2BCHE
SCHEMBL7809943 0.83 CNR2 (0.33) CNR2BCHEACHE
SCHEMBL7817393 0.81 KDM4E (0.35) NQO2NQO1CYP19A1RAD52MEN1
SCHEMBL7817848 0.80 TOP2A (0.40) NQO1CNR2BCHEACHE
SCHEMBL7808985 0.79 TOP2A (0.40) NQO2NQO1KAT2BSMARCA2KEAP1
SCHEMBL7804639 0.75 ECE1 (0.40) NQO2NQO1KAT2BATMEHMT2
SCHEMBL7805085 0.75 ECE1 (0.40) KAT2BEHMT2
SCHEMBL9389199 0.75 TOP2A (0.40) CYP19A1MEN1KMT2AEHMT2
SCHEMBL7809049 0.74 EHMT2 (0.39) NQO2NQO1KAT2BEHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750619-B1 HETERO-ANNULATED INDAZOLES NOVUSPHARMA SPA (IT) 2001-05-30 EP disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed