SCHEMBL7809943

SCHEMBL7809943

COc1ccc(COc2cncc3c2-c2nn(C)c4ccc(Cl)c(c24)C3=O)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.33
CNR1 P21554 1/20 0.33
KDM4E B2RXH2 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
NPBWR1 P48145 2/20 0.33
P2RX7 Q99572 1/20 0.32
TOP2A P11388 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MCHR1 Q99705 1/20 0.32
PPARG P37231 1/20 0.32
CHRM5 P08912 1/20 0.32
FGFR1 P11362 1/20 0.32
SRC P12931 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817848 0.87 TOP2A (0.40) CNR2CNR1KDM4ECYP1A2CYP2C9
SCHEMBL7819175 0.83 NQO2 (0.39) CNR2BCHEACHE
SCHEMBL7821575 0.81 TOP2A (0.35) CNR2TOP2ASRCBCHE
SCHEMBL7819169 0.77 KDM4E (0.36) KDM4ECYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL7817393 0.72 KDM4E (0.35) KDM4ECYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL7809332 0.68 TDP2 (0.45) TOP2A
SCHEMBL10806544 0.67 MAPK13 (0.62) KDM4ECYP1A2ALDH1A1TOP2A
SCHEMBL6829824 0.64 NPC1 (0.45) KDM4ECYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL10799732 0.64 MAPK13 (0.38) KDM4EALDH1A1LMNAPOLBCYP3A4
SCHEMBL2434210 0.63 NPBWR1 (0.44) KDM4EALDH1A1LMNAPOLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750619-B1 HETERO-ANNULATED INDAZOLES NOVUSPHARMA SPA (IT) 2001-05-30 EP disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
EP-0750619-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA S.p.A. (IT) 1997-01-02 EP disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed