SCHEMBL7817848

SCHEMBL7817848

COc1ccc(COc2cncc3c2-c2nn(CCN(C)C)c4ccc(Cl)c(c24)C3=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 12/20 0.40
CNR2 P34972 3/20 0.37
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.36
NQO1 P15559 1/20 0.36
KCNH2 Q12809 1/20 0.34
MCHR1 Q99705 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
CNR1 P21554 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7818284 0.87 NQO2 (0.38) TOP2ACNR2BCHEACHENQO1
SCHEMBL7809943 0.87 CNR2 (0.33) TOP2ACNR2BCHEACHEMCHR1
SCHEMBL7821158 0.85 TOP2A (0.35) TOP2ACNR2BCHEACHENQO1
SCHEMBL7821575 0.83 TOP2A (0.35) TOP2ACNR2BCHESMN1; SMN2
SCHEMBL7819175 0.80 NQO2 (0.39) CNR2BCHEACHENQO1
SCHEMBL7804662 0.75 TOP2A (0.48) TOP2AKCNH2SMN1; SMN2KDM4ECYP3A4
SCHEMBL7817393 0.75 KDM4E (0.35) NQO1SMN1; SMN2KDM4ELMNACYP1A2
SCHEMBL7819985 0.73 TOP2A (0.51) TOP2A
SCHEMBL7819169 0.72 KDM4E (0.36) TOP2AKDM4ELMNACYP1A2POLB
SCHEMBL7812061 0.69 TOP2A (0.45) TOP2ANQO1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750619-B1 HETERO-ANNULATED INDAZOLES NOVUSPHARMA SPA (IT) 2001-05-30 EP disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
EP-0750619-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA S.p.A. (IT) 1997-01-02 EP disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed