SCHEMBL7821158

SCHEMBL7821158

COc1ccc(COc2cncc3c2-c2nn(CCN(C)C)c4ccc(NCCN)c(c24)C3=O)cc1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 8/20 0.35
CNR2 P34972 2/20 0.34
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
NQO2 P16083 3/20 0.33
NQO1 P15559 2/20 0.33
IGF1R P08069 1/20 0.32
KCNH2 Q12809 1/20 0.32
MCHR1 Q99705 1/20 0.32
BRD4 O60885 1/20 0.31
ECE1 P42892 1/20 0.31
MUS81 Q96NY9 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7818284 0.95 NQO2 (0.38) TOP2ACNR2BCHEACHENQO2
SCHEMBL7819175 0.88 NQO2 (0.39) CNR2BCHEACHENQO2NQO1
SCHEMBL7817848 0.85 TOP2A (0.40) TOP2ACNR2BCHEACHENQO1
SCHEMBL7818947 0.81 TOP2A (0.44) TOP2ANQO2NQO1ECE1MUS81
SCHEMBL7822606 0.80 TOP2A (0.36) TOP2ACNR2BCHEBRD4
SCHEMBL7804809 0.78 ECE1 (0.47) TOP2AECE1MUS81SMN1; SMN2
SCHEMBL7804602 0.78 ECE1 (0.47) TOP2AECE1MUS81
SCHEMBL7817109 0.76 TOP2A (0.44) TOP2A
SCHEMBL7809103 0.75 TOP2A (0.46) TOP2ANQO2NQO1SMN1; SMN2
SCHEMBL7809335 0.74 TOP2A (0.44) TOP2ANQO2NQO1ECE1MUS81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750619-B1 HETERO-ANNULATED INDAZOLES NOVUSPHARMA SPA (IT) 2001-05-30 EP disclosed
EP-0775143-A1 NEW 3-SUBSTITUTED 3H-2,3-BENZODIAZEPINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-28 EP disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
EP-0750619-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA S.p.A. (IT) 1997-01-02 EP disclosed
WO-1996004283-A1 NEW 3-SUBSTITUTED 3H-2,3-BENZODIAZEPINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS SCHERING AKTIENGESELLSCHAFT (DE) 1996-02-15 WO disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed