SCHEMBL7819214

SCHEMBL7819214

COc1ccc(-c2cnc(SCC(=O)NC(Cc3ccc(Cl)c(Cl)c3)C3CCNC3)nc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.42
GRIN1 Q05586 2/20 0.37
GRIN2B Q13224 2/20 0.37
IKBKB O14920 1/20 0.37
TP53 P04637 2/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SSTR3 P32745 1/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
MAPT P10636 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
MEN1 O00255 1/20 0.35
APOBEC3A P31941 1/20 0.35
KMT2A Q03164 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MMP1 P03956 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7830259 0.99 AKT1 (0.41) AKT1GRIN1GRIN2BIKBKBTP53
SCHEMBL6028207 0.95 CHEK1 (0.39) AKT1GRIN1GRIN2BIKBKBTP53
SCHEMBL6029095 0.89 CHEK1 (0.39) GRIN1GRIN2BTP53LMNAMAPT
SCHEMBL6028748 0.89 CHEK1 (0.39) GRIN1GRIN2BTP53LMNAMAPT
SCHEMBL7829880 0.87 AKT1 (0.42) AKT1GRIN1GRIN2BIKBKBSSTR3
SCHEMBL7819254 0.87 MCHR1 (0.43) TP53LMNAMAPTMEN1KMT2A
SCHEMBL6029187 0.87 MAPT (0.38) GRIN1GRIN2BTP53LMNAMAPT
SCHEMBL7828843 0.87 AKT1 (0.42) AKT1GRIN1GRIN2BIKBKBSSTR3
Hydrochloric Acid SCHEMBL7833338 0.87 AKT1 (0.42) AKT1GRIN1GRIN2BIKBKBSSTR3
SCHEMBL7830301 0.87 AKT1 (0.44) AKT1GRIN1GRIN2BIKBKBSSTR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131288-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-09-12 EP disclosed
WO-2000031032-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO disclosed