SCHEMBL7828843

SCHEMBL7828843

COc1ccc(-c2cnc(NCC(=O)NC(Cc3ccc(Cl)c(Cl)c3)C3CCNC3)nc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.42
HSP90AA1 P07900 1/20 0.40
SCD O00767 3/20 0.39
CLK4 Q9HAZ1 2/20 0.38
CLK1 P49759 1/20 0.38
CLK2 P49760 1/20 0.38
DYRK1A Q13627 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
GRIN1 Q05586 2/20 0.37
GRIN2B Q13224 2/20 0.37
IKBKB O14920 1/20 0.37
CHEK1 O14757 1/20 0.36
SSTR3 P32745 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7829880 0.88 AKT1 (0.42) AKT1HSP90AA1SCDCLK4CLK1
Hydrochloric Acid SCHEMBL7833338 0.87 AKT1 (0.42) AKT1HSP90AA1SCDCLK4CLK1
SCHEMBL7830301 0.87 AKT1 (0.44) AKT1HSP90AA1SCDGRIN1GRIN2B
SCHEMBL7819214 0.87 AKT1 (0.42) AKT1HSP90AA1GRIN1GRIN2BIKBKB
Hydrochloric Acid SCHEMBL7830259 0.86 AKT1 (0.41) AKT1HSP90AA1GRIN1GRIN2BIKBKB
SCHEMBL7819177 0.84 CNR2 (0.44) AKT1SSTR3SLC6A2SLC6A4SLC6A3
SCHEMBL6029151 0.83 CHEK1 (0.39) AKT1SCDCLK4CLK1CLK2
SCHEMBL6028846 0.83 AKT1 (0.40) AKT1GRIN1GRIN2BCHEK1SSTR3
SCHEMBL6028207 0.82 CHEK1 (0.39) AKT1GRIN1GRIN2BIKBKBCHEK1
SCHEMBL7827088 0.79 DYRK1A (0.39) AKT1CLK4DYRK1AIKBKBJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131288-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-09-12 EP disclosed
WO-2000031032-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO disclosed