SCHEMBL7830301

SCHEMBL7830301

COc1ccc(-c2cnc(CCC(=O)NC(Cc3ccc(Cl)c(Cl)c3)C3CCNC3)nc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.44
GRIN1 Q05586 4/20 0.37
GRIN2B Q13224 4/20 0.37
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MMP7 P09237 1/20 0.37
MMP9 P14780 1/20 0.37
MMP8 P22894 1/20 0.37
MMP13 P45452 1/20 0.37
SSTR3 P32745 1/20 0.36
ALDH1A1 P00352 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FLT3 P36888 1/20 0.36
P2RX7 Q99572 1/20 0.35
SCD O00767 1/20 0.35
IKBKB O14920 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6028846 0.95 AKT1 (0.40) AKT1GRIN1GRIN2BSSTR3ALDH1A1
SCHEMBL7833614 0.91 AKT1 (0.38) AKT1SLC6A2SLC6A4SLC6A3IKBKB
SCHEMBL7829880 0.88 AKT1 (0.42) AKT1GRIN1GRIN2BMMP1MMP2
Hydrochloric Acid SCHEMBL7833338 0.87 AKT1 (0.42) AKT1GRIN1GRIN2BMMP1MMP2
SCHEMBL7828843 0.87 AKT1 (0.42) AKT1GRIN1GRIN2BMMP1MMP2
SCHEMBL7819214 0.87 AKT1 (0.42) AKT1GRIN1GRIN2BMMP1MMP2
SCHEMBL6029616 0.86 CDK2 (0.37) AKT1
Hydrochloric Acid SCHEMBL7830259 0.86 AKT1 (0.41) AKT1GRIN1GRIN2BMMP1MMP2
SCHEMBL7818522 0.85 SLC6A4 (0.38) AKT1GRIN1GRIN2BMMP1MMP2
SCHEMBL6029125 0.85 MAPK1 (0.38) AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131288-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-09-12 EP disclosed
WO-2000031032-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO disclosed