SCHEMBL7829880

SCHEMBL7829880

COc1ccc(-c2cnc(OCC(=O)NC(Cc3ccc(Cl)c(Cl)c3)C3CCNC3)nc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.42
GRIN1 Q05586 2/20 0.38
GRIN2B Q13224 2/20 0.38
IKBKB O14920 1/20 0.37
CTSD P07339 1/20 0.37
CLK4 Q9HAZ1 2/20 0.37
CLK1 P49759 1/20 0.37
CLK2 P49760 1/20 0.37
DYRK1A Q13627 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
SSTR3 P32745 1/20 0.37
SCD O00767 3/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
MMP1 P03956 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7833338 0.99 AKT1 (0.42) AKT1GRIN1GRIN2BIKBKBCTSD
SCHEMBL6029151 0.95 CHEK1 (0.39) AKT1GRIN1GRIN2BIKBKBCLK4
SCHEMBL7827088 0.91 DYRK1A (0.39) AKT1IKBKBCLK4DYRK1ASLC6A2
SCHEMBL7830301 0.88 AKT1 (0.44) AKT1GRIN1GRIN2BIKBKBSSTR3
SCHEMBL7828843 0.88 AKT1 (0.42) AKT1GRIN1GRIN2BIKBKBCLK4
SCHEMBL7819214 0.87 AKT1 (0.42) AKT1GRIN1GRIN2BIKBKBSSTR3
SCHEMBL6030392 0.87 CHEK1 (0.41) AKT1GRIN1GRIN2BCLK4CLK1
Hydrochloric Acid SCHEMBL7830259 0.87 AKT1 (0.41) AKT1GRIN1GRIN2BIKBKBSSTR3
SCHEMBL6029200 0.86 ROCK2 (0.38) AKT1IKBKBCLK4DYRK1AROCK2
SCHEMBL7826595 0.85 SLC6A4 (0.39) AKT1GRIN1GRIN2BCTSDSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131288-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-09-12 EP disclosed
WO-2000031032-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO disclosed