SCHEMBL7821785

SCHEMBL7821785

Nc1nc(-c2ccc3c(c2)CCC3)nc2nc[nH]c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLA1 P09884 1/20 0.46
PDPK1 O15530 1/20 0.45
GDA Q9Y2T3 1/20 0.45
ADORA3 P0DMS8 13/20 0.43
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ADORA1 P30542 11/20 0.41
ADORA2A P29274 4/20 0.40
ADORA2B P29275 3/20 0.40
PIK3CA P42336 3/20 0.40
PIK3CG P48736 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7830739 0.80 PDPK1 (0.41) POLA1PDPK1GDAADORA3ADORA1
Hydrochloric Acid SCHEMBL7832921 0.79 PDPK1 (0.40) POLA1PDPK1GDAADORA3ADORA1
SCHEMBL7821784 0.79 ALDH1A1 (0.42) POLA1MEN1NPC1ALDH1A1TP53
SCHEMBL7830814 0.77 NEK2 (0.48) PDPK1GDAALDH1A1MAPTSMN1; SMN2
SCHEMBL7833385 0.76 MPO (0.45) POLA1PDPK1GDA
Hydrochloric Acid SCHEMBL7833212 0.76 NEK2 (0.48) PDPK1GDAALDH1A1MAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL7834487 0.75 MPO (0.44) POLA1PDPK1GDA
SCHEMBL1741361 0.74 ADORA3 (0.69) PDPK1GDAADORA3ADORA1ADORA2A
SCHEMBL29791254 0.74 ADORA3 (0.69) PDPK1GDAADORA3ADORA1ADORA2A
SCHEMBL7249956 0.73 BRAF (0.50) PDPK1GDAADORA3ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP claimed
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP disclosed