SCHEMBL7822145

SCHEMBL7822145

COC(=O)c1c(C)c(C)cc2nc(OC)c(OC)nc12

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
ALDH1A1 P00352 6/20 0.40
KDM4E B2RXH2 5/20 0.40
HPGD P15428 5/20 0.40
CYP3A4 P08684 2/20 0.40
ACHE P22303 1/20 0.38
POLB P06746 2/20 0.38
ATM Q13315 2/20 0.36
CISD2 Q8N5K1 1/20 0.36
CASP1 P29466 1/20 0.36
HSD17B10 Q99714 1/20 0.36
DHODH Q02127 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7825789 0.82 CSNK2A1 (0.40) ALDH1A1KDM4EHPGDCYP3A4ACHE
SCHEMBL7592279 0.81 SMN1; SMN2 (0.38) GAAALDH1A1KDM4EHPGDCYP3A4
SCHEMBL7470942 0.72 L3MBTL1 (0.37) GAAALDH1A1KDM4EHPGDACHE
SCHEMBL7810829 0.72 NQO2 (0.33) POLB
SCHEMBL7468982 0.71 ALDH1A1 (0.45) GAAALDH1A1KDM4EHPGDCYP3A4
SCHEMBL22690002 0.69 POLB (0.50) GAAALDH1A1KDM4EHPGDCYP3A4
SCHEMBL7811964 0.69 NQO2 (0.33) POLB
SCHEMBL7472004 0.69 ALDH1A1 (0.36) GAAALDH1A1KDM4EHPGDCYP3A4
SCHEMBL7598494 0.68 KMT2A (0.38) ALDH1A1CYP3A4POLBMEN1KMT2A
SCHEMBL27459361 0.68 NQO2 (0.48) GAAALDH1A1KDM4ECYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781279-B1 QUINOXALINEDIONE NMDA RECEPTOR ANTAGONISTS PFIZER LTD (GB) 2001-06-13 EP disclosed
US-5783572-A TREATMENT OF NEURODEGENERATIVE DISORDERS PFIZER INC. (US) 1998-07-21 US disclosed
EP-0781279-A1 QUINOXALINEDIONE NMDA RECEPTOR ANTAGONISTS Pfizer Limited (GB) 1997-07-02 EP disclosed
WO-1996008485-A1 QUINOXALINEDIONE NMDA RECEPTOR ANTAGONISTS PFIZER LIMITED (GB) 1996-03-21 WO disclosed