SCHEMBL7472004

SCHEMBL7472004

CCS(=O)(=O)Nc1c(C)c(C)cc2nc(OC)c(OC)nc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
GAA P10253 1/20 0.36
NPY1R P25929 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LY6K Q17RY6 1/20 0.35
HPGD P15428 5/20 0.35
LMNA P02545 2/20 0.35
HSD17B10 Q99714 1/20 0.35
CREBBP Q92793 3/20 0.32
KDM4E B2RXH2 2/20 0.32
NPC1 O15118 1/20 0.32
HTT P42858 1/20 0.32
MAPT P10636 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
RECQL P46063 1/20 0.32
CRHR1 P34998 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468982 0.86 ALDH1A1 (0.45) ALDH1A1GAANPY1RSMN1; SMN2HPGD
SCHEMBL7476854 0.82 PTGS1 (0.37) ALDH1A1GAANPY1RSMN1; SMN2
SCHEMBL7462801 0.80 CCR4 (0.36) SMN1; SMN2LY6KHPGDLMNAHSD17B10
SCHEMBL7467654 0.74 NPY1R (0.37) ALDH1A1GAANPY1RSMN1; SMN2HSD17B10
SCHEMBL7476942 0.73 ALDH1A1 (0.38) ALDH1A1GAANPY1RSMN1; SMN2HPGD
SCHEMBL7822145 0.69 GAA (0.40) ALDH1A1GAASMN1; SMN2HPGDHSD17B10
SCHEMBL7465420 0.68 SMN1; SMN2 (0.33) ALDH1A1GAANPY1RSMN1; SMN2LMNA
SCHEMBL7470942 0.68 L3MBTL1 (0.37) ALDH1A1GAASMN1; SMN2HPGDLMNA
SCHEMBL7810829 0.68 NQO2 (0.33) LMNANPC1MAPTRECQL
SCHEMBL7811964 0.68 NQO2 (0.33) LMNANPC1MAPTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0783495-B1 QUINOXALINE DERIVATIVES USEFUL IN THERAPY PFIZER LTD (GB) 2002-02-27 EP disclosed
US-5852016-A Quinoxaline derivatives useful in therapy PFIZER INC. (US) 1998-12-22 US disclosed
WO-1996009295-A1 QUINOXALINE DERIVATIVES USEFUL IN THERAPY PFIZER LIMITED (GB) 1996-03-28 WO disclosed