SCHEMBL7825860

SCHEMBL7825860

CC(C)(NC(=O)c1ccc(C#N)cc1)C(C(=O)O)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 4/20 0.58
CTSG P08311 4/20 0.58
CTRB1 P17538 4/20 0.58
CMA1 P23946 4/20 0.58
S1PR4 O95977 2/20 0.46
S1PR3 Q99500 2/20 0.46
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
SLC6A9 P48067 1/20 0.44
SLC6A5 Q9Y345 1/20 0.44
EPHX2 P34913 3/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
TMEM97 Q5BJF2 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837285 0.89 EPHX2 (0.55) PRSS1CTSGCTRB1CMA1CYP2C9
SCHEMBL7838715 0.89 PRSS1 (0.46) PRSS1CTSGCTRB1CMA1S1PR4
SCHEMBL7836737 0.87 PRSS1 (0.48) PRSS1CTSGCTRB1CMA1S1PR4
SCHEMBL7826105 0.87 MEN1 (0.52) PRSS1CTSGCTRB1CMA1S1PR4
SCHEMBL7836194 0.87 PRSS1 (0.47) PRSS1CTSGCTRB1CMA1EPHX2
SCHEMBL7835566 0.84 PRSS1 (0.45) PRSS1CTSGCTRB1CMA1S1PR4
SCHEMBL7835765 0.81 MEN1 (0.49) PRSS1CTSGCTRB1CMA1EPHX2
SCHEMBL7837405 0.78 MEN1 (0.47) PRSS1CTSGCTRB1CMA1EPHX2
SCHEMBL7837709 0.77 EPHX2 (0.47) PRSS1CTSGCTRB1CMA1EPHX2
SCHEMBL7834153 0.77 PRSS1 (0.45) PRSS1CTSGCTRB1CMA1S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed