SCHEMBL7835765

SCHEMBL7835765

CC(C(=O)O)C(C)(C)NC(=O)c1ccc(C#N)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
PRSS1 P07477 4/20 0.47
CTSG P08311 4/20 0.47
CTRB1 P17538 4/20 0.47
CMA1 P23946 4/20 0.47
EPHX2 P34913 3/20 0.47
TRPA1 O75762 1/20 0.43
ALDH1A1 P00352 1/20 0.43
PKM P14618 1/20 0.43
MLYCD O95822 1/20 0.43
GSK3B P49841 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PPARA Q07869 1/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837405 0.86 MEN1 (0.47) MEN1KMT2APRSS1CTSGCTRB1
SCHEMBL7837709 0.82 EPHX2 (0.47) MEN1KMT2APRSS1CTSGCTRB1
SCHEMBL7825860 0.81 PRSS1 (0.58) MEN1KMT2APRSS1CTSGCTRB1
SCHEMBL7825622 0.80 NPC1 (0.46) MEN1KMT2APRSS1CTSGCTRB1
SCHEMBL7837208 0.80 CTSG (0.47) MEN1KMT2APRSS1CTSGCTRB1
SCHEMBL507273 0.79 EPHX2 (0.55) MEN1KMT2APRSS1CTSGCTRB1
SCHEMBL7837285 0.78 EPHX2 (0.55) MEN1KMT2APRSS1CTSGCTRB1
SCHEMBL7835600 0.78 CTSG (0.46) MEN1KMT2APRSS1CTSGCTRB1
SCHEMBL7838715 0.78 PRSS1 (0.46) MEN1KMT2APRSS1CTSGCTRB1
SCHEMBL7826783 0.77 CTSG (0.47) MEN1KMT2APRSS1CTSGCTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed