SCHEMBL7836737

SCHEMBL7836737

CC(C)(NC(=O)c1ccc(C#N)cc1)C(C(=O)O)c1cccc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 4/20 0.48
CTSG P08311 4/20 0.48
CTRB1 P17538 4/20 0.48
CMA1 P23946 4/20 0.48
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
SLC6A9 P48067 1/20 0.43
SLC6A5 Q9Y345 1/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
TRPA1 O75762 3/20 0.39
S1PR3 Q99500 3/20 0.39
S1PR4 O95977 2/20 0.39
S1PR1 P21453 2/20 0.38
S1PR5 Q9H228 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7825860 0.87 PRSS1 (0.58) PRSS1CTSGCTRB1CMA1CYP2D6
SCHEMBL7826105 0.82 MEN1 (0.52) PRSS1CTSGCTRB1CMA1CYP2D6
SCHEMBL7837285 0.79 EPHX2 (0.55) PRSS1CTSGCTRB1CMA1CYP2C9
SCHEMBL7838715 0.79 PRSS1 (0.46) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL7836741 0.78 PRSS1 (0.62) PRSS1CTSGCTRB1CMA1CYP2D6
SCHEMBL7837372 0.78 ITGB3 (0.45) PRSS1CTSGCTRB1CMA1CYP2D6
SCHEMBL7836194 0.77 PRSS1 (0.47) PRSS1CTSGCTRB1CMA1CYP3A4
SCHEMBL7835566 0.77 PRSS1 (0.45) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL7835765 0.74 MEN1 (0.49) PRSS1CTSGCTRB1CMA1MEN1
SCHEMBL5947886 0.74 EPHX2 (0.63) CYP2D6CYP2C9SLC6A9SLC6A5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed