SCHEMBL7826151

SCHEMBL7826151

O=C1CN(c2ccccc2)C(=O)N1C(=O)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.71
RAB9A P51151 3/20 0.71
KMT2A Q03164 3/20 0.71
MEN1 O00255 2/20 0.58
CTSG P08311 9/20 0.48
CMA1 P23946 9/20 0.48
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
CDK2 P24941 1/20 0.43
PDE5A O76074 1/20 0.42
P2RX4 Q99571 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836516 0.91 KMT2A (0.60) NPC1RAB9AKMT2AMEN1CTSG
SCHEMBL7838574 0.89 KMT2A (0.58) NPC1RAB9AKMT2AMEN1CTSG
SCHEMBL7837364 0.85 KMT2A (0.55) NPC1RAB9AKMT2AMEN1CTSG
SCHEMBL7837528 0.84 TSHR (0.53) NPC1RAB9AKMT2AMEN1CTSG
SCHEMBL7838811 0.83 NPC1 (1.00) NPC1RAB9AKMT2AMEN1CTSG
SCHEMBL7837470 0.83 CTSG (0.53) NPC1RAB9AKMT2AMEN1CTSG
SCHEMBL7836895 0.82 KMT2A (0.51) NPC1RAB9AKMT2AMEN1CTSG
SCHEMBL7833371 0.82 CTSG (0.54) NPC1RAB9AKMT2ACTSGCMA1
SCHEMBL921684 0.81 NPC1 (0.51) NPC1RAB9AKMT2AMEN1CTSG
SCHEMBL7835354 0.80 CTSG (0.51) NPC1RAB9AKMT2AMEN1CTSG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721944-B1 IMIDAZOLIDINE DERIVATIVE AND USE THEREOF SUNTORY LTD (JP) 2001-01-17 EP disclosed
US-5691335-A CARDIOVASCULAR DISORDERS SUNTORY LIMITED (JP) 1997-11-25 US disclosed
EP-0721944-A1 IMIDAZOLIDINE DERIVATIVE AND USE THEREOF SUNTORY LIMITED (JP) 1996-07-17 EP disclosed