SCHEMBL7827129

SCHEMBL7827129

N#CCC(C=O)(c1ccccc1)c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.34
DRD2 P14416 2/20 0.33
DRD4 P21917 2/20 0.33
OPRM1 P35372 2/20 0.33
DRD3 P35462 2/20 0.33
CYP2D6 P10635 2/20 0.33
KIF11 P52732 1/20 0.33
CYP3A4 P08684 1/20 0.32
ALDH1A1 P00352 5/20 0.32
TSHR P16473 4/20 0.32
MAPT P10636 1/20 0.31
HTT P42858 2/20 0.31
CYP2C19 P33261 1/20 0.31
HIF1A Q16665 1/20 0.31
KCNA3 P22001 1/20 0.30
KCNN4 O15554 1/20 0.30
MCL1 Q07820 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7816528 0.81 MAPT (0.35) ATMDRD2DRD4OPRM1DRD3
SCHEMBL8992344 0.80 TSHR (0.34) ATMALDH1A1TSHRHTTCYP2C19
SCHEMBL8891559 0.78 MAPT (0.39) CYP3A4ALDH1A1MAPT
SCHEMBL8891565 0.78 MAPT (0.39) CYP3A4ALDH1A1MAPT
SCHEMBL1148767 0.77 KCNN4 (0.40) ATMDRD2OPRM1DRD3KIF11
SCHEMBL27379002 0.77 ALDH1A1 (0.38) CYP2D6ALDH1A1TSHRMAPTHTT
SCHEMBL6311548 0.72 ALDH1A1 (0.38) CYP3A4ALDH1A1TSHRHTTCYP2C19
SCHEMBL342226 0.72 ALDH1A1 (0.38) DRD2OPRM1DRD3CYP3A4ALDH1A1
SCHEMBL27880149 0.72 ALDH1A1 (0.38) ALDH1A1TSHRHTTCYP2C19HIF1A
SCHEMBL10587806 0.72 ATM (0.39) ATMDRD2DRD4OPRM1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712845-B1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-17 EP disclosed
WO-1997024325-A1 DIPHENYLMETHANE DERIVATIVES AS MIP-1α/RANTES RECEPTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-10 WO disclosed
US-5633248-A GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS, DIARYLALKYLIDENEDIAMINES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-27 US disclosed
EP-0712845-A1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-22 EP disclosed