SCHEMBL7828183

SCHEMBL7828183

CCOC(=O)C(Cc1ccc([N+](=O)[O-])cc1[N+](=O)[O-])C(=O)OCC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.54
TDP1 Q9NUW8 3/20 0.54
CYP1A2 P05177 1/20 0.54
MAPT P10636 8/20 0.52
MAPK1 P28482 5/20 0.52
SMN1; SMN2 Q16637 5/20 0.52
L3MBTL1 Q9Y468 4/20 0.50
LMNA P02545 3/20 0.50
KMT2A Q03164 3/20 0.50
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
KDM4E B2RXH2 2/20 0.49
GAA P10253 2/20 0.48
MITF O75030 1/20 0.46
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
MTOR P42345 1/20 0.44
RAB9A P51151 1/20 0.44
TP53 P04637 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18371949 0.88 MAPT (0.46) ALDH1A1TDP1CYP1A2MAPTMAPK1
SCHEMBL28216693 0.85 ALDH1A1 (0.52) ALDH1A1TDP1MAPTMAPK1SMN1; SMN2
SCHEMBL17049174 0.84 MAPT (0.55) ALDH1A1TDP1MAPTMAPK1SMN1; SMN2
SCHEMBL9834203 0.83 ALDH1A1 (0.47) ALDH1A1TDP1MAPTMAPK1SMN1; SMN2
SCHEMBL28260499 0.83 MAPT (0.47) ALDH1A1TDP1MAPTMAPK1SMN1; SMN2
SCHEMBL22165764 0.83 MAPT (0.49) ALDH1A1TDP1MAPTMAPK1SMN1; SMN2
SCHEMBL27956774 0.82 HPD (0.48) ALDH1A1CYP1A2MAPTMAPK1L3MBTL1
SCHEMBL1572954 0.82 L3MBTL1 (0.56) ALDH1A1MAPTMAPK1SMN1; SMN2L3MBTL1
SCHEMBL30619954 0.82 L3MBTL1 (0.56) ALDH1A1MAPTMAPK1SMN1; SMN2L3MBTL1
SCHEMBL18371980 0.82 MAPT (0.44) ALDH1A1TDP1MAPTMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329389-B1 HETEROCYCLIC AMINES AND DERIVATIVES, SOMATOSTATIN AND ANTIDIABETIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-12-11 US disclosed
EP-1070054-A1 AMINE COMPOUNDS, THEIR PRODUCTION AND THEIR USE AS SOMATOSTATIN RECEPTOR ANTAGONISTS OR AGONISTS Takeda Chemical Industries, Ltd. (JP) 2001-01-24 EP disclosed
WO-1999052875-A1 AMINE COMPOUNDS, THEIR PRODUCTION AND THEIR USE AS SOMATOSTATIN RECEPTOR ANTAGONISTS OR AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-21 WO disclosed