SCHEMBL7828184

SCHEMBL7828184

Clc1cccc(Cl)c1CBr.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.48
CYP3A4 P08684 1/20 0.48
AKR1B1 P15121 1/20 0.39
ESR1 P03372 2/20 0.39
ESR2 Q92731 2/20 0.39
TAAR1 Q96RJ0 2/20 0.38
DPP4 P27487 1/20 0.37
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 1/20 0.35
TSHR P16473 3/20 0.35
LMNA P02545 1/20 0.35
TRPA1 O75762 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
ATM Q13315 1/20 0.33
KMT2A Q03164 1/20 0.32
GAA P10253 1/20 0.32
FEN1 P39748 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9770 0.82 TAAR1 (0.50) CYP3A4AKR1B1TAAR1DPP4ALDH1A1
SCHEMBL11029873 0.80 TAAR1 (0.48) CYP3A4AKR1B1TAAR1DPP4ALDH1A1
SCHEMBL5356053 0.75 TDP1 (0.67) TDP1CYP3A4ESR1ESR2ALDH1A1
Dibromomethane SCHEMBL7950072 0.75 TDP1 (0.75) TDP1CYP3A4ESR1ESR2ALDH1A1
Dibromomethane SCHEMBL5329477 0.75 TDP1 (0.75) TDP1CYP3A4ESR1ESR2ALDH1A1
SCHEMBL9804209 0.73 CYP3A4 (0.50) TDP1CYP3A4ESR1ESR2ALDH1A1
1,2-Dibromoethane SCHEMBL28837174 0.73 TDP1 (0.71) TDP1CYP3A4ESR1ESR2ALDH1A1
1,4-Dichlorobenzene SCHEMBL11803922 0.73 CYP3A4 (0.71) TDP1CYP3A4ESR1ESR2ALDH1A1
SCHEMBL28407819 0.72 CYP3A4 (0.52) TDP1CYP3A4AKR1B1ESR1ESR2
Benzyl Bromide SCHEMBL1043932 0.72 TSHR (0.70) TDP1CYP3A4ESR1ESR2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757682-B1 BENZOFURAN DERIVATIVES USEFUL AS INHIBITORS OF BONE RESORPTION FUJISAWA PHARMACEUTICAL CO (JP) 2001-06-20 EP disclosed
EP-0757682-A1 BENZOFURAN DERIVATIVES USEFUL AS INHIBITORS OF BONE RESORPTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed