SCHEMBL7828371

SCHEMBL7828371

COc1ccc2c(c1)CCC1(CCCCN1)C2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.59
SMN1; SMN2 Q16637 1/20 0.40
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
DRD5 P21918 1/20 0.40
DRD3 P35462 1/20 0.40
KDM1A O60341 1/20 0.40
POLA1 P09884 2/20 0.40
PRNP P04156 1/20 0.39
ADRB2 P07550 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2B P18089 1/20 0.39
SLC6A2 P23975 1/20 0.39
HTR2C P28335 1/20 0.39
HRH1 P35367 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39
HTR2B P41595 1/20 0.39
HTR5A P47898 1/20 0.39
SLC6A3 Q01959 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7822802 0.99 ADRA2A (0.57) ADRA2ASMN1; SMN2DRD2DRD1DRD5
Hydrochloric Acid SCHEMBL7816122 0.99 ADRA2A (0.57) ADRA2ASMN1; SMN2DRD2DRD1DRD5
Hydrochloric Acid SCHEMBL7827227 0.99 ADRA2A (0.57) ADRA2ASMN1; SMN2DRD2DRD1DRD5
Hydrochloric Acid SCHEMBL7831175 0.84 ADRA2A (0.43) ADRA2ASMN1; SMN2ADRA2BHRH1
SCHEMBL9049906 0.80 ADRA2A (0.55) ADRA2ASMN1; SMN2DRD2DRD1DRD5
Hydrochloric Acid SCHEMBL7815957 0.80 ALDH1A1 (0.49) ADRA2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL7826706 0.79 ADRA2A (0.54) ADRA2ASMN1; SMN2DRD2DRD1DRD5
Hydrochloric Acid SCHEMBL29051753 0.78 ADRA2A (0.56) ADRA2ADRD2DRD1DRD5DRD3
Hydrochloric Acid SCHEMBL30468426 0.78 ADRA2A (0.56) ADRA2ADRD2DRD1DRD5DRD3
Hydrochloric Acid SCHEMBL8841918 0.77 DRD2 (0.38) ADRA2ADRD2DRD1DRD5DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712845-B1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-17 EP disclosed
US-5633248-A GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS, DIARYLALKYLIDENEDIAMINES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-27 US disclosed
EP-0712845-A1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-22 EP disclosed
EP-0670313-A1 Spiro compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-09-06 EP disclosed