SCHEMBL78287

SCHEMBL78287

O=C(NN=Cc1ccccc1)C(=O)NN=Cc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 1.00
KMT2A Q03164 6/20 1.00
RAB9A P51151 5/20 0.61
SMN1; SMN2 Q16637 3/20 0.59
NPC1 O15118 3/20 0.59
G6PD P11413 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
CTRC Q99895 1/20 0.58
ALDH1A1 P00352 2/20 0.58
NOX4 Q9NPH5 1/20 0.56
LMNA P02545 2/20 0.56
HDAC3 O15379 1/20 0.56
HDAC2 Q92769 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
NCOR2 Q9Y618 1/20 0.56
MAPT P10636 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9067815 1.00 MEN1 (1.00) MEN1KMT2ARAB9ASMN1; SMN2NPC1
SCHEMBL549490 1.00 MEN1 (1.00) MEN1KMT2ARAB9ASMN1; SMN2NPC1
SCHEMBL333482 1.00 MEN1 (1.00) MEN1KMT2ARAB9ASMN1; SMN2NPC1
SCHEMBL5081924 0.91 MEN1 (0.82) MEN1KMT2ARAB9ASMN1; SMN2NPC1
SCHEMBL5081918 0.91 MEN1 (0.82) MEN1KMT2ARAB9ASMN1; SMN2NPC1
SCHEMBL4115183 0.87 MEN1 (0.77) MEN1KMT2ARAB9ASMN1; SMN2NPC1
SCHEMBL4115180 0.87 MEN1 (0.77) MEN1KMT2ARAB9ASMN1; SMN2NPC1
SCHEMBL31588094 0.87 MEN1 (0.77) MEN1KMT2ARAB9ASMN1; SMN2NPC1
Phenylsemicarbazone SCHEMBL11882629 0.83 MEN1 (0.71) MEN1KMT2ARAB9ASMN1; SMN2NPC1
SCHEMBL13496984 0.83 MEN1 (0.71) MEN1KMT2ARAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3933 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2920236-B1 POLYMER COMPOSITION HAVING IMPROVED LONG-TERM STABILITY, MOULDED PARTS PRODUCED THEREFROM AND INTENDED USES THEREOF FRAUNHOFER GES FORSCHUNG (DE) 2019-06-05 EP claimed
US-9856364-B2 Stabilized reversible polymer composition XEROX CORPORATION (US) 2018-01-02 US claimed
EP-3166999-A1 THERMAL INTERFACE MATERIAL WITH ION SCAVENGER Honeywell International Inc. (US) 2017-05-17 EP claimed
US-20160272789-A1 POLYMER COMPOSITION WITH IMPROVED LONG-TERM STABILITY, MOULDED PARTS PRODUCED HEREFROM AND ALSO PURPOSES OF USE FRAUNHOFER-GESELLACHAFT ZUR FÖRDERUNG DER ANGEWANDTEN FORSCHUNG E.V. (DE) 2016-09-22 US claimed
WO-2016004565-A1 THERMAL INTERFACE MATERIAL WITH ION SCAVENGER HONEYWELL INTERNATIONAL INC. (US) 2016-01-14 WO claimed
EP-2920236-A1 POLYMER COMPOSITION HAVING IMPROVED LONG-TERM STABILITY, MOULDED PARTS PRODUCED THEREFROM AND INTENDED USES THEREOF FRAUNHOFER-GESELLSCHAFT zur Förderung der angewandten Forschung e.V. (DE) 2015-09-23 EP claimed
US-20140353549-A1 STABILIZED REVERSIBLE POLYMER COMPOSITION XEROX CORPORATION (US) 2014-12-04 US claimed
WO-2014076273-A1 POLYMER COMPOSITION HAVING IMPROVED LONG-TERM STABILITY, MOULDED PARTS PRODUCED THEREFROM AND INTENDED USES THEREOF Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2014-05-22 WO claimed
CN-101942142-B Preparation method of semiconductive shielding material for 110kV and above voltage class cables JIANGYIN HAIJIANG POLYMER MATERIAL CO LTD 2012-08-15 CN claimed
US-7951859-B2 Composition with enhanced heat resistance property UNION CARBIDE CHEMICALS & PLASTICS TECHNOLOGY LLC (US) 2011-05-31 US claimed
WO-1990002770-A2 AQUEOUS ADDITIVE SYSTEMS, METHODS AND POLYMERIC PARTICLES EASTMAN KODAK COMPANY (US) 1990-03-22 WO claimed
WO-1989011502-A1 AQUEOUS ADDITIVE SYSTEMS, METHODS AND POLYMERIC PARTICLES EASTMAN KODAK COMPANY (US) 1989-11-30 WO claimed
EP-0142467-B1 POLYMER COMPOUNDS CONTAINING PIPERIDYL GROUPS AND THEIR USE AS STABILISERS IN SYNTHETIC POLYMERS CIBA-GEIGY S.p.A. (IT) 1988-08-24 EP claimed
EP-0140297-A2 Thiocarbamic-acid esters as stabilizers CIBA-GEIGY AG (CH) 1985-05-08 EP claimed
EP-0070168-B1 PROTECTING METAL SUBSTRATES FROM CORROSION RAYCHEM CORPORATION (a California corporation) (US) 1985-04-10 EP claimed
US-4455204-A ADHESIVES RAYCHEM CORPORATION (US) 1984-06-19 US claimed
EP-0108714-A1 Dibenzodioxaphosphepine and dioxaphosphocine processing stabilizers CIBA-GEIGY AG (CH) 1984-05-16 EP claimed
EP-0006418-B1 PREVENTION OF PVC POLYMER BUILDUP IN POLYMERIZATION REACTORS USING OXALYL BIS(BENZYLIDENEHYDRAZIDE) AND ALUMINA Conoco Phillips Company (US) 1983-03-09 EP claimed
EP-0006418-A1 Prevention of PVC polymer buildup in polymerization reactors using oxalyl bis(benzylidenehydrazide) and alumina Conoco Phillips Company (US) 1980-01-09 EP claimed
US-4145496-A Prevention of PVC polymer buildup in polymerization reactors using oxalyl bis(benzylidenehydrazide) and alumina CONTINENTAL OIL COMPANY (US) 1979-03-20 US claimed