SCHEMBL7828783

SCHEMBL7828783

CN(C)c1ncc(-c2cccc(Nc3ccc(-c4ccco4)cc3[N+](=O)[O-])c2)cn1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.41
POLB P06746 3/20 0.40
MAPT P10636 4/20 0.39
RXFP1 Q9HBX9 1/20 0.39
ALK Q9UM73 1/20 0.38
EGFR P00533 1/20 0.36
ERN1 O75460 1/20 0.36
AKR1B10 O60218 1/20 0.36
AKR1B1 P15121 1/20 0.36
AKR1C4 P17516 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7831824 0.88 TP53 (0.41) TP53POLBMAPTRXFP1ALK
SCHEMBL7834274 0.86 AKR1B1 (0.36) POLBMAPTERN1AKR1B10AKR1B1
SCHEMBL2643726 0.84 ALK (0.42) ALKEGFR
Fluoride SCHEMBL27482913 0.81 L3MBTL1 (0.39) POLBMAPTEGFRAKR1B10AKR1B1
SCHEMBL5755261 0.79 L3MBTL1 (0.39) POLBMAPTAKR1B10AKR1B1AKR1C4
SCHEMBL7834286 0.74 ALK (0.46) ALKEGFR
SCHEMBL2643906 0.74 TP53 (0.41) TP53POLBMAPTRXFP1ALK
SCHEMBL7820330 0.73 MAPT (0.40) POLBMAPTERN1AKR1B10AKR1B1
SCHEMBL7820033 0.72 ABL1 (0.44) TP53POLBMAPTRXFP1ALK
Fluoride SCHEMBL2643534 0.68 MAPT (0.42) POLBMAPTAKR1B10AKR1B1AKR1C4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1164134-A1 Benzimidazole compounds and their use as modulators of the GABA A receptor complex NEUROSEARCH A/S (DK) 2001-12-19 EP disclosed
EP-0751133-B1 Pyrimidine compound, and liquid crystal composition and liquid crystal element using the same MITSUI CHEMICALS INC (JP) 2001-09-12 EP disclosed
US-5922724-A Benzimidazole compounds and their use as modulators of the GABA a receptor complex NEUROSEARCH A/S (DK) 1999-07-13 US disclosed
US-5770108-A HIGH SPEED RESPONSE, MOLECULAR ORIENTATION, HIGH CONTRAST, RECEPTIVITY MITSUI TOATSU CHEMICALS, INC. (JP) 1998-06-23 US disclosed
EP-0751133-A1 Pyrimidine compound, and liquid crystal composition and liquid crystal element using the same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1997-01-02 EP disclosed