SCHEMBL7829063

SCHEMBL7829063

[CH]=CC(=O)c1ccccc1Cl

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.58
CES1 P23141 1/20 0.58
ALDH1A1 P00352 1/20 0.56
POLB P06746 2/20 0.52
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47
CYP1A2 P05177 2/20 0.46
HPGD P15428 2/20 0.46
CYP2C19 P33261 1/20 0.46
ERCC5 P28715 1/20 0.44
FEN1 P39748 1/20 0.44
RAB9A P51151 1/20 0.43
TP53 P04637 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TSHR P16473 1/20 0.42
RECQL P46063 1/20 0.42
SMO Q99835 2/20 0.41
CXCL12 P48061 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL293634 0.80 CES2 (0.60) CES2CES1ALDH1A1POLBPTGS1
SCHEMBL29952517 0.80 CES2 (0.60) CES2CES1ALDH1A1POLBPTGS1
Water SCHEMBL10353121 0.78 CES2 (0.58) CES2CES1ALDH1A1POLBPTGS1
SCHEMBL4770585 0.78 CES2 (0.58) CES2CES1ALDH1A1POLBPTGS1
SCHEMBL9113114 0.78 CES2 (0.58) CES2CES1ALDH1A1POLBPTGS1
SCHEMBL7006496 0.78 CES2 (0.58) CES2CES1ALDH1A1POLBPTGS1
SCHEMBL15563306 0.78 ALDH1A1 (0.55) CES2CES1ALDH1A1POLBPTGS1
SCHEMBL15563304 0.78 ALDH1A1 (0.55) CES2CES1ALDH1A1POLBPTGS1
SCHEMBL7830798 0.76 KDM4E (0.55) ALDH1A1PTGS1PTGS2HPGDCYP2C19
SCHEMBL18334775 0.75 CES2 (0.54) CES2CES1ALDH1A1POLBPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686636-B1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA CO (JP) 2001-04-04 EP disclosed
US-5840895-A INTERMEDIATES FOR ANTIALLERGENS MEIJI SEIKA KABUSHIKI KAISHA (JP) 1998-11-24 US disclosed
US-5686442-A ANTIALLERGENS MEIJI SEIKA KABUSHIKI KAISHA (JP) 1997-11-11 US disclosed
EP-0686636-A1 TRICYCLIC BENZAZEPINE AND BENZOTHIAZEPINE DERIVATIVES MEIJI SEIKA KABUSHIKI KAISHA (JP) 1995-12-13 EP disclosed