SCHEMBL7829191

SCHEMBL7829191

CCOC(=O)C=Cc1c(C)oc2c(NC(=O)c3c(Cl)cccc3Cl)cccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.47
L3MBTL1 Q9Y468 2/20 0.45
LMNA P02545 4/20 0.43
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
MDM2 Q00987 1/20 0.42
ALDH1A1 P00352 2/20 0.41
TDP1 Q9NUW8 1/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
POLB P06746 2/20 0.38
HTT P42858 2/20 0.37
GPR35 Q9HC97 1/20 0.37
GHSR Q92847 1/20 0.37
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9272800 1.00 MAPT (0.47) MAPTL3MBTL1LMNAMEN1KMT2A
SCHEMBL7828330 0.81 KMT2A (0.43) MAPTLMNAMEN1KMT2AALDH1A1
SCHEMBL7829801 0.80 KMT2A (0.41) MAPTLMNAMEN1KMT2AALDH1A1
SCHEMBL6537907 0.79 MAPT (0.44) MAPTL3MBTL1LMNAMEN1KMT2A
SCHEMBL6537905 0.79 MAPT (0.44) MAPTL3MBTL1LMNAMEN1KMT2A
SCHEMBL7832320 0.79 MAPT (0.42) MAPTLMNAMEN1KMT2AALDH1A1
SCHEMBL7823933 0.78 MAPT (0.48) MAPTLMNAMEN1KMT2AALDH1A1
SCHEMBL8341922 0.78 GPR35 (0.42) MAPTLMNAMEN1KMT2AALDH1A1
SCHEMBL8926694 0.78 MEN1 (0.54) MAPTL3MBTL1LMNAMEN1KMT2A
SCHEMBL7817291 0.77 RAB9A (0.41) MAPTLMNAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757682-B1 BENZOFURAN DERIVATIVES USEFUL AS INHIBITORS OF BONE RESORPTION FUJISAWA PHARMACEUTICAL CO (JP) 2001-06-20 EP disclosed
EP-0757682-A1 BENZOFURAN DERIVATIVES USEFUL AS INHIBITORS OF BONE RESORPTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-12 EP disclosed
WO-1995029907-A1 BENZOFURAN DERIVATIVES USEFUL AS INHIBITORS OF BONE RESORPTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-09 WO disclosed