SCHEMBL7829318

SCHEMBL7829318

O=C(O)Cc1nc(-c2cc3ccccc3o2)no1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 2/20 0.46
PDE4B Q07343 1/20 0.44
PDE4D Q08499 1/20 0.44
ALDH1A1 P00352 5/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
KDM4E B2RXH2 5/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MMP12 P39900 1/20 0.42
MMP13 P45452 1/20 0.42
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 1/20 0.41
GAA P10253 1/20 0.41
NFKB1 P19838 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837657 0.87 ALDH1A1 (0.53) PSMB5ALDH1A1MEN1KMT2ATSHR
SCHEMBL7818703 0.85 ALDH1A1 (0.64) PSMB5ALDH1A1MEN1KMT2ARAB9A
SCHEMBL7829263 0.80 HPGD (0.46) PSMB5ALDH1A1KMT2AMAPK1HPGD
SCHEMBL4611029 0.76 ALDH1A1 (0.68) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL4034138 0.70 NPC1 (0.65) ALDH1A1NPC1RAB9ATSHRKDM4E
SCHEMBL7829321 0.70 AKR1B1 (0.46) ALDH1A1KDM4EHPGDTDP1MCL1
SCHEMBL30561833 0.70 MAOB (0.55) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL11555365 0.70 AKR1B1 (0.51) ALDH1A1KMT2ATSHRSMN1; SMN2MAPT
SCHEMBL4400216 0.70 ALDH1A1 (0.58) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL1650806 0.70 ESR1 (0.57) PSMB5ALDH1A1MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329389-B1 HETEROCYCLIC AMINES AND DERIVATIVES, SOMATOSTATIN AND ANTIDIABETIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-12-11 US disclosed
EP-1070054-A1 AMINE COMPOUNDS, THEIR PRODUCTION AND THEIR USE AS SOMATOSTATIN RECEPTOR ANTAGONISTS OR AGONISTS Takeda Chemical Industries, Ltd. (JP) 2001-01-24 EP disclosed
WO-1999052875-A1 AMINE COMPOUNDS, THEIR PRODUCTION AND THEIR USE AS SOMATOSTATIN RECEPTOR ANTAGONISTS OR AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-21 WO disclosed