SCHEMBL7829429

SCHEMBL7829429

O=C(O)c1cc2cc(OCc3ccccc3)ccc2n1S(=O)(=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.66
MCL1 Q07820 2/20 0.64
BCL2 P10415 1/20 0.64
BID P55957 1/20 0.64
SRD5A2 P31213 2/20 0.57
HDAC1 Q13547 2/20 0.47
LTB4R Q15722 1/20 0.47
LTB4R2 Q9NPC1 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
MRGPRX4 Q96LA9 1/20 0.47
ABCB11 O95342 2/20 0.46
BCL2L1 Q07817 1/20 0.45
PPARG P37231 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SRD5A1 P18405 1/20 0.42
ACLY P53396 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6598140 0.91 CCR2 (0.54) CCR2MCL1BCL2BIDSRD5A2
SCHEMBL31159405 0.88 BCL2 (0.66) CCR2MCL1BCL2BIDSRD5A2
SCHEMBL6543181 0.82 MCL1 (0.59) CCR2MCL1BCL2BIDSRD5A2
SCHEMBL20761835 0.82 BCL2 (0.58) MCL1BCL2BIDSRD5A2HDAC1
SCHEMBL6596517 0.81 CCR2 (0.73) CCR2MCL1BCL2BIDABCB11
SCHEMBL6542672 0.80 BCL2 (0.59) CCR2MCL1BCL2BIDSRD5A2
SCHEMBL7638737 0.80 BCL2 (0.59) CCR2MCL1BCL2BIDSRD5A2
SCHEMBL6959828 0.80 CCR2 (1.00) CCR2MCL1BCL2BIDHDAC1
SCHEMBL20742924 0.80 SRD5A2 (0.60) MCL1BCL2BIDSRD5A2HDAC1
SCHEMBL6953098 0.79 CCR2 (0.75) CCR2MCL1BCL2BIDABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150952-A1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 RECEPTOR ANTAGONISTS AstraZeneca AB (SE) 2001-11-07 EP disclosed
WO-2000046196-A1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS ASTRAZENECA AB (SE) 2000-08-10 WO disclosed