SCHEMBL7829477

SCHEMBL7829477

O=c1[nH]c2c(O)ccc(CCNCCCS(=O)(=O)CCNCCc3ccccc3)c2s1

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 18/20 0.81
ADRB1 P08588 3/20 0.81
ABCB11 O95342 2/20 0.81
DRD2 P14416 2/20 0.81
PDE4A P27815 1/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7842790 0.99 ADRB2 (0.80) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL7839897 0.91 ABCB11 (0.77) ADRB2ADRB1ABCB11DRD2PDE4A
Hydrochloric Acid SCHEMBL7839511 0.90 ABCB11 (0.76) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL8528403 0.90 ABCB11 (0.93) ADRB2ADRB1ABCB11DRD2PDE4A
Sibenadet SCHEMBL30438496 0.90 ADRB2 (1.00) ADRB2ADRB1ABCB11DRD2PDE4A
Sibenadet SCHEMBL48983 0.90 ADRB2 (1.00) ADRB2ADRB1ABCB11DRD2PDE4A
Sibenadet SCHEMBL249498 0.89 ADRB2 (0.98) ADRB2ADRB1ABCB11DRD2PDE4A
Hydrochloric Acid SCHEMBL8527365 0.89 ABCB11 (0.92) ADRB2ADRB1ABCB11DRD2PDE4A
Sibenadet SCHEMBL678828 0.88 ADRB2 (0.97) ADRB2ADRB1ABCB11DRD2PDE4A
Hydrochloric Acid SCHEMBL8899662 0.85 ADRB2 (0.63) ADRB2ADRB1ABCB11DRD2PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558677-B1 BIOLOGICALLY ACTIVE AMINES ASTRAZENECA AB (SE) 2001-08-16 EP claimed
US-5648370-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1997-07-15 US claimed
EP-0558677-A1 BIOLOGICALLY ACTIVE AMINES Astra Pharmaceuticals Limited (GB) 1993-09-08 EP claimed
WO-1992008708-A1 BIOLOGICALLY ACTIVE AMINES FISONS PLC (GB) 1992-05-29 WO claimed