SCHEMBL7829503

SCHEMBL7829503

CC1(C)OC=C(c2ccncc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.40
DRD2 P14416 6/20 0.36
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
CDC7 O00311 5/20 0.33
ROCK1 Q13464 4/20 0.33
DBF4 Q9UBU7 4/20 0.33
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33
TP53 P04637 1/20 0.32
PKM P14618 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7832946 0.80 CYP2A6 (0.44) SIGMAR1MAPTLMNATP53
SCHEMBL7830887 0.70 KDM4E (0.42) MAPTLMNATP53PKM
SCHEMBL7829992 0.69 SIGMAR1 (0.47) SIGMAR1DRD2MAPTLMNAPTGS2
SCHEMBL286590 0.68 KMT2A (0.35) MAPTLMNACDC7ROCK1DBF4
SCHEMBL30267491 0.64 PIK3CD (0.46) MAPTCDC7PIK3CDPIK3CAPIK3CB
SCHEMBL12189104 0.64 TP53 (0.34) MAPTLMNACDC7ROCK1DBF4
SCHEMBL286625 0.63 SIGMAR1 (0.36) SIGMAR1DRD2MAPTLMNACDC7
SCHEMBL21316072 0.62 MAPT (0.50) MAPTLMNATP53PKM
SCHEMBL15000221 0.61 RAB9A (0.40) LMNACDC7TP53PTGS2
SCHEMBL1003235 0.60

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105125547-A FORUM PHARMACEUTICALS INC FORUM PHARMACEUTICALS INC 2015-12-09 CN disclosed
CN-102459242-B Phenoxymethyl heterocyclic compounds FORUM PHARMACEUTICALS INC. (US) 2015-08-26 CN disclosed
EP-1109799-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-27 EP disclosed
WO-2000061571-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-10-19 WO disclosed