SCHEMBL7829992

SCHEMBL7829992

CC1(C)OC=C(c2ccc3ccccc3c2)C1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.47
DRD2 P14416 2/20 0.47
GSTP1 P09211 1/20 0.44
PTGER3 P43115 6/20 0.43
LPL P06858 1/20 0.42
LIPG Q9Y5X9 1/20 0.42
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
NOTUM Q6P988 1/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
HDAC4 P56524 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
ACMSD Q8TDX5 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27468872 0.79 SIGMAR1 (0.57) SIGMAR1DRD2
SCHEMBL11479263 0.76 SIGMAR1 (0.44) SIGMAR1DRD2GSTP1PTGER3
SCHEMBL28042699 0.73 BACE1 (0.50) SIGMAR1DRD2HPGDKDM4EMAPT
SCHEMBL11314945 0.73 DRD2 (0.42) SIGMAR1DRD2GSTP1PTGER3LMNA
SCHEMBL7832796 0.71 PTGS2 (0.40) PTGS1PTGS2HDAC4HDAC2HDAC8
SCHEMBL7829503 0.69 SIGMAR1 (0.40) SIGMAR1DRD2LMNAMAPTPTGS2
SCHEMBL3646655 0.67 GSTP1 (0.52) GSTP1PTGER3ALDH1A1KDM4ENOTUM
SCHEMBL4269525 0.66 GSTP1 (0.42) SIGMAR1DRD2GSTP1PTGER3LPL
SCHEMBL5013872 0.65 ESR1 (0.71) GSTP1ALDH1A1KDM4EMAPTACMSD
SCHEMBL15902840 0.65 ESR1 (0.71) GSTP1ALDH1A1KDM4EMAPTACMSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-27 EP disclosed
WO-2000061571-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-10-19 WO disclosed