SCHEMBL7829574

SCHEMBL7829574

O=C1C=c2cc(COc3ncnc4ncccc34)ccc2=N1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.36
CDC7 O00311 3/20 0.33
DBF4 Q9UBU7 3/20 0.33
KDR P35968 1/20 0.33
RXFP1 Q9HBX9 3/20 0.31
ALDH1A1 P00352 2/20 0.30
NPC1 O15118 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30
EGFR P00533 1/20 0.30
MAPT P10636 1/20 0.30
PKM P14618 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837582 0.81 EGFR (0.35) KDRNPC1EGFRMAPT
SCHEMBL7838604 0.80 EGFR (0.35) LMNAKDRRXFP1ALDH1A1EGFR
SCHEMBL8813155 0.73 NPC1 (0.32) ALDH1A1NPC1CYP2C19EGFR
SCHEMBL7822327 0.72 RXRB (0.41) LMNACDC7DBF4ALDH1A1NPC1
SCHEMBL8815271 0.72 F2 (0.36) ALDH1A1NPC1MAPTMEN1KMT2A
SCHEMBL7829575 0.72 MAOB (0.47) LMNAKDR
SCHEMBL7347464 0.65 TOP1 (0.49) NPC1MEN1KMT2A
SCHEMBL5485288 0.65 NPC1 (0.38) LMNAALDH1A1NPC1EGFRMAPT
SCHEMBL9430440 0.64 HCAR2 (0.48) NPC1MEN1KMT2A
SCHEMBL9792739 0.63 CYP11B1 (0.41) LMNANPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP claimed